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Phage-encoded combinatorial chemical libraries based on bicyclic peptides
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Nature chemical biology, 2011-03, Vol.7 (3), p.174-181
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Family-wide chemical profiling and structural analysis of PARP and tankyrase inhibitors
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Acetylation site specificities of lysine deacetylase inhibitors in human cells
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Small-molecule inhibition of APT1 affects Ras localization and signaling
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Halofuginone and other febrifugine derivatives inhibit prolyl-tRNA synthetase
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The Design of Covalent Allosteric Drugs
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Crystal structures of oseltamivir-resistant influenza virus neuraminidase mutants
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VX-680, a potent and selective small-molecule inhibitor of the Aurora kinases, suppresses tumor growth in vivo
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Histone deacetylase inhibitors reverse gene silencing in Friedreich's ataxia
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